AR - androgen receptor | Elisa - Clia - Antibody - Protein

Family main features

Background

The androgen receptor (AR) is a type of nuclear receptor that is activated by binding to androgens, which are male sex hormones such as testosterone and dihydrotestosterone (DHT). AR plays a pivotal role in the development and maintenance of male characteristics and reproductive activity. It is also involved in various other physiological processes, including muscle growth, bone density maintenance, and certain behaviors. AR dysfunction or mutations can lead to a range of disorders, including androgen insensitivity syndrome, prostate cancer, and other androgen-related conditions.


Protein Structure

AR is composed of several distinct domains:

  • N-terminal Domain (NTD): Contains the activation function-1 (AF-1) region, which is responsible for transcriptional activation. This domain is highly variable and essential for interaction with co-regulators.
  • DNA-binding Domain (DBD): Composed of two zinc finger motifs, this domain binds to specific DNA sequences known as androgen response elements (AREs) in the promoter regions of target genes.
  • Hinge Region: Provides flexibility and contains a nuclear localization signal essential for the receptor's transport into the nucleus.
  • Ligand-binding Domain (LBD): Binds androgens and contains the activation function-2 (AF-2) region. This domain is crucial for receptor dimerization and interaction with heat shock proteins and co-regulators.


Classification and Subtypes

AR is a member of the nuclear receptor subfamily 3, group C (NR3C4). Unlike some other nuclear receptors, AR does not have subtypes but exists in multiple isoforms resulting from alternative splicing and post-translational modifications.


Function and Biological Significance

AR mediates the effects of androgens by regulating the expression of specific genes:

  • Sexual Development: Essential for the development of male genitalia and secondary sexual characteristics during puberty.
  • Reproductive Function: Influences spermatogenesis and fertility.
  • Muscle and Bone Health: Promotes muscle mass and strength, and supports bone density.
  • Behavioral Effects: Involved in the regulation of libido and other androgen-influenced behaviors.


Clinical Issues

  • Prostate Cancer: AR signaling is a major driver of prostate cancer progression. Therapeutic strategies often target AR to inhibit its activity in advanced prostate cancer.
  • Androgen Insensitivity Syndrome (AIS): Mutations in the AR gene can lead to partial or complete insensitivity to androgens, resulting in a spectrum of phenotypes from mild undervirilization to complete feminization.
  • Spinal and Bulbar Muscular Atrophy (SBMA): Also known as Kennedy's disease, is a neurodegenerative disorder caused by a mutation in the AR gene.


Summary

The androgen receptor (AR) is a critical nuclear receptor that mediates the biological effects of androgens, influencing male development, reproductive functions, muscle and bone health, and certain behaviors. Its structure includes domains essential for androgen binding, DNA interaction, and transcriptional regulation. Dysregulation or mutations in AR can lead to conditions like prostate cancer, androgen insensitivity syndrome, and spinal and bulbar muscular atrophy, making it a significant target for clinical research and therapeutic interventions.

AR Recommended name:

androgen receptor (AR)

Aliases for AR

KD,AIS,AR8,TFM,DHTR,SBMA,HYSP1,NR3C4,SMAX1,HUMARA,Dihydrotestosterone receptor,Nuclear receptor subfamily 3 group C member 4

En la tabla siguiente se muestra una comparativa de todos los reactivos disponibles en nuestro catálogo (Proteins and Peptides, ELISA Kits, Primary Antibodies, CLIA Kits, Antibody Pairs) relacionados con AR - androgen receptor

Se muestran ordenados por categorías para poder comparar cómodamente sus características principales. Esta tabla, que contiene un enlace con la ficha de cada producto, es exportable a Excel.

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immunoassays

providerCodereferencenamereactivitysample typeassay typetest rangesensitivitypricesize 1uniprot idstatus
AbbexaARabx516031Dog Androgen Receptor (AR) ELISA KitDogTissue homogenates, cell lysates and other biological fluids.0.156 ng/ml - 10 ng/ml71596 testsQ9TT90RUO
FineTestAREH0033Human AR(Androgen receptor) ELISA KithumanSerum,Plasma,Tissue homogenates,Other biological fluidsSandwich ELISA, Double Antibody0.313-20ng/ml96TP10275RUO
AbbexaARabx572052Human Testosterone Receptor (AR) ELISA KitHumanTissue homogenates, cell lysates and other biological fluids.Sandwich78 pg/ml - 5000 pg/ml46.9 pg/ml61196 testsP10275RUO
AbbexaARabx492549Human Androgen Receptor (AR) CLIA KitHumanTissue homogenates, cell lysates and other biological fluids.Sandwich0.312 ng/ml - 20 ng/ml< 0.113 ng/ml84596 testsRUO
AbbexaARabx250172Human Androgen Receptor (AR) ELISA KitHumanTissue homogenates, cell lysates and other biological fluids.Sandwich0.312 ng/ml - 20 ng/ml0.19 ng/ml61196 testsP10275RUO
AbbexaARabx595032Androgen Receptor Cell ELISA KitHuman513.596 testsP10275RUO
AbbexaARabx150644Human Androgen Receptor (AR) ELISA KitHumanTissue homogenates, cell lysates and other biological fluids.Sandwich0.312 ng/ml - 20 ng/ml< 0.12 ng/ml68996 testsRUO
AbbexaARabx196434Human Androgen Receptor (AR) CLIA KitHumanSerum, plasma and other biological fluids.Sandwich78 pg/ml - 5000 pg/ml46.9 pg/ml643.596 testsRUO
AbbexaARabx596601Androgen Receptor (pS650) DNA-Binding ELISA KitHuman58596 testsP10275RUO
AbbexaARabx596602Androgen Receptor (pY363) DNA-Binding ELISA KitHuman58596 testsP10275RUO
AbbexaARabx596463Androgen Receptor DNA-Binding ELISA KitHuman55996 testsP10275RUO
AbbexaARabx596067Androgen Receptor (pY363) Cell ELISA KitHuman5462 × 96 testsP10275RUO
AbbexaARabx360101Monkey Androgen Receptor (AR) ELISA KitMonkeySerum, plasma and other biological fluids.Sandwich31.2 pg/ml - 2000 pg/ml18.8 pg/ml68996 testsRUO
AbbexaARabx492550Mouse Androgen Receptor (AR) CLIA KitMouseTissue homogenates, cell lysates and other biological fluids.Sandwich0.156 ng/ml - 10 ng/ml< 0.055 ng/ml84596 testsRUO
AbbexaARabx153631Mouse Androgen Receptor (AR) ELISA KitMouseTissue homogenates, cell lysates, cell culture supernatants and other biological fluids.Sandwich0.156 ng/ml - 10 ng/ml< 0.06 ng/ml643.596 testsRUO
AbbexaARabx361833Pig Androgen Receptor (AR) ELISA KitPigTissue homogenates, cell lysates, cell culture supernatant and other biological fluids.Sandwich31.2 pg/ml - 2000 pg/ml18.8 pg/ml71596 testsRUO
AbbexaARabx362258Rabbit Androgen Receptor (AR) ELISA KitRabbitSerum, plasma and other biological fluids.Sandwich0.312 ng/ml - 20 ng/ml0.19 ng/ml68996 testsRUO
AbbexaARabx155192Rat Androgen Receptor (AR) ELISA KitRatTissue homogenates, cell lysates and other biological fluids.Sandwich0.156 ng/ml - 10 ng/ml< 0.07 ng/ml643.596 testsRUO
AbbexaARabx492551Rat Androgen Receptor (AR) CLIA KitRatTissue homogenates, cell lysates, cell culture supernatants and other biological fluids.Sandwich0.156 ng/ml - 10 ng/ml< 0.059 ng/ml84596 testsRUO

Primary Antibodies

providerCodereferencenamereactivityclonalityhostimmunogen targetisotypeconjugationtested applicationspricesize 1uniprot idstatus
AbbexaARabx341269Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB16920 µlP10275RUO
AbbexaARabx431104Androgen Receptor (AR) AntibodyHumanPolyclonalGoatAndrogen Receptor (AR)IgGUnconjugatedP-ELISA, WB, IHC, IF/ICC416200 µlRUO
AbbexaARabx011627Androgen Receptor (AR) AntibodyHumanMonoclonalMouseAndrogen Receptor (AR)IgG1UnconjugatedELISA383.5100 µlP10275RUO
AbbexaARabx011626Androgen Receptor (AR) AntibodyHumanMonoclonalMouseAndrogen Receptor (AR)IgG1UnconjugatedELISA, WB, IHC383.5100 µlP10275RUO
AbbexaARabx313222Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, IHC16920 µgP10275RUO
AbbexaARabx171210Androgen Receptor (AR) AntibodyHumanMonoclonalMouseAndrogen Receptor (AR)UnconjugatedWB, IHC, IF/ICC7801 mlRUO
AbbexaARabx402159Androgen Receptor (AR) AntibodyHumanMonoclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, IHC29950 µlP10275RUO
AbbexaARabx313225Androgen Receptor (AR) Antibody (Biotin)HumanPolyclonalRabbitAndrogen Receptor (AR)IgGBiotinELISA16920 µgP10275RUO
AbbexaARabx000354AR (pS213) AntibodyHumanPolyclonalRabbitAR (pS213)IgGUnconjugatedWB20820 µlP10275RUO
AbbexaARabx322922Androgen Receptor Phospho-Ser650 (AR pS650) AntibodyHumanPolyclonalRabbitAndrogen Receptor Phospho-Ser650 (AR pS650)IgGUnconjugatedELISA, IHC22150 µgP10275RUO
AbbexaARabx272116Androgen Receptor (AR) Antibody (Biotin)HumanPolyclonalRabbitAndrogen Receptor (AR)IgGBiotinWB, IHC, IF/ICC364200 µlRUO
AbbexaARabx025510Androgen Receptor Protein (AR) AntibodyHumanMonoclonalMouseAndrogen Receptor Protein (AR)IgAUnconjugatedELISA, WB292.580 µlP10275RUO
AbbexaARabx313223Androgen Receptor (AR) Antibody (HRP)HumanPolyclonalRabbitAndrogen Receptor (AR)IgGHRPELISA16920 µgP10275RUO
AbbexaARabx313224Androgen Receptor (AR) Antibody (FITC)HumanPolyclonalRabbitAndrogen Receptor (AR)IgGFITC16920 µgP10275RUO
AbbexaARabx324576Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB, IHC22150 µgP10275RUO
AbbexaARabx339753Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, IHC26050 µlP10275RUO
AbbexaARabx000355AR (pS650) AntibodyHumanPolyclonalRabbitAR (pS650)IgGUnconjugatedELISA20820 µlP10275RUO
AbbexaARabx377564Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB, IHC26050 µgP10275RUO
AbbexaARabx322977Androgen Receptor Phospho-Ser213 (AR pS213) AntibodyHumanPolyclonalRabbitAndrogen Receptor Phospho-Ser213 (AR pS213)IgGUnconjugatedELISA, IHC22150 µgP10275RUO
AbbexaARabx322976Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, IHC22150 µgP10275RUO
AbbexaARabx332866Androgen Receptor Phospho-Ser213 (AR pS213) AntibodyHumanPolyclonalRabbitAndrogen Receptor Phospho-Ser213 (AR pS213)IgGUnconjugatedELISA, WB, IF/ICC429100 µlP10275RUO
AbbexaARabx341157Androgen Receptor (AR) AntibodyHumanMonoclonalMouseAndrogen Receptor (AR)IgG2b KappaUnconjugatedELISA, IHC26050 µlP10275RUO
AbbexaARabx402119Androgen Receptor (AR) AntibodyHumanMonoclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB, IHC29950 µlP10275RUO
AbbexaARabx101255Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)UnconjugatedWB, IHC, IF/ICC273100 µlP10275RUO
AbbexaARabx332994Androgen Receptor Phospho-Ser650 (AR pS650) AntibodyHumanPolyclonalRabbitAndrogen Receptor Phospho-Ser650 (AR pS650)IgGUnconjugatedELISA, WB, IHC429100 µlP10275RUO
AbbexaARabx325329Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, IHC, IF/ICC22150 µgP10275RUO
AbbexaARabx325135Androgen Receptor Phospho-Ser94 (AR pS94) AntibodyHumanPolyclonalRabbitAndrogen Receptor Phospho-Ser94 (AR pS94)IgGUnconjugatedELISA, IF/ICC22150 µgP10275RUO
AbbexaARabx025053Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB, IHC292.580 µlP10275RUO
AbbexaARabx012943Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB5210 µgP10275RUO
AbbexaARabx327189Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB22150 µgP10275RUO
AbbexaARabx327037Androgen Receptor Phospho-Tyr363 (AR pY363) AntibodyHumanPolyclonalRabbitAndrogen Receptor Phospho-Tyr363 (AR pY363)IgGUnconjugatedELISA, WB22150 µgP10275RUO
AbbexaARabx148286Androgen Receptor Phospho-Tyr534 (AR pY534) AntibodyHumanPolyclonalRabbitAndrogen Receptor Phospho-Tyr534 (AR pY534)UnconjugatedWB31250 µlP10275RUO
AbbexaARabx001670Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedWB31260 µlP10275RUO
AbbexaARabx117188Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB, IHC, IF/ICC468100 µlP10275RUO
AbbexaARabx327348Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB22150 µgP10275RUO
AbbexaARabx012635Androgen Receptor (Phospho-Tyr363) AntibodyHumanPolyclonalRabbitAndrogen ReceptorIgGUnconjugatedELISA, WB5210 µgP10275RUO
AbbexaARabx038452Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB357.5100 µgRUO
AbbexaARabx011629Androgen Receptor (AR) AntibodyHumanPolyclonalRabbitAndrogen Receptor (AR)IgGUnconjugatedELISA, WB, IHC364100 µgP10275RUO
AbbexaARabx101254Androgen Receptor (AR) AntibodyMousePolyclonalRabbitAndrogen Receptor (AR)UnconjugatedWB, IHC, IF/ICC273100 µlP19091RUO
AbbexaARabx101256Androgen Receptor (AR) AntibodyRatPolyclonalRabbitAndrogen Receptor (AR)UnconjugatedWB, IHC, IF/ICC286100 µlP15207RUO
AbbexaARabx101257Androgen Receptor (AR) AntibodyRatPolyclonalRabbitAndrogen Receptor (AR)UnconjugatedWB, IHC, IF/ICC286100 µlP15207RUO
AbbexaARabx131716Androgen Receptor (AR) AntibodyRatMonoclonalMouseAndrogen Receptor (AR)IgG2b KappaUnconjugatedWB, IHC, IF/ICC299100 µlP15207RUO
AbbexaARabx273243Androgen Receptor (AR) Antibody (Biotin)RatPolyclonalRabbitAndrogen Receptor (AR)IgGBiotinWB, IHC, IF/ICC390200 µlRUO
AbbexaARabx132571Androgen Receptor (AR) AntibodyRatMonoclonalMouseAndrogen Receptor (AR)IgGUnconjugatedWB, IHC, IF/ICC299100 µlRUO

Proteins and Peptides

providerCodereferencenameoriginexpressionhostconjugationtested applicationspricesize 1uniprot idstatus
AbbexaARabx269552Androgen Receptor (AR) PeptideSyntheticUnconjugatedP-ELISA175.5100 µg
AbbexaARabx065299Human Androgen Receptor (AR) ProteinHumanRecombinantE. coliUnconjugatedWB, SDS-PAGE22110 µgP10275RUO
AbbexaARabx065301Rat Androgen Receptor (AR) ProteinRatRecombinantE. coliUnconjugatedWB, SDS-PAGE28991 mgP15207RUO
FineTestARP8071Recombinant Human ARHumanRecombinantE.ColiWestern Blot, ELISA50μgP10275RUO
AbbexaARabx065302Mouse Androgen Receptor (AR) ProteinMouseRecombinantE. coliUnconjugatedWB, SDS-PAGE23410 µgP19091RUO
AbbexaARabx065300Rat Androgen Receptor (AR) ProteinRatRecombinantE. coliUnconjugatedWB, SDS-PAGE26010 µgP15207RUO
FineTestARP0503Recombinant Human ARHumanRecombinantE.ColiWestern Blot, ELISA50μgP10275RUO

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